VUF 10166

CAS No. 155584-74-0

VUF 10166 ( —— )

Catalog No. M17335 CAS No. 155584-74-0

VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 37 In Stock
10MG 59 In Stock
25MG 112 In Stock
100MG 299 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    VUF 10166
  • Note
    Research use only, not for human use.
  • Brief Description
    VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.
  • Description
    VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.
  • Synonyms
    ——
  • Pathway
    Angiogenesis
  • Target
    EGFR
  • Recptor
    5-HT3A; 5-HT3AB
  • Research Area
    Inflammation/Immunology
  • Indication
    ——

Chemical Information

  • CAS Number
    155584-74-0
  • Formula Weight
    262.74
  • Molecular Formula
    C13H15ClN4
  • Purity
    98%
  • Solubility
    ——
  • SMILES
    CN1CCN(CC1)C1=NC2=CC=CC=C2N=C1Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Thompson AJ, et al. J Pharmacol Exp Ther, 2012, 341(2), 350-9.
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