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VUF 10166
CAS No. 155584-74-0
VUF 10166( —— )
Catalog No. M17335 CAS No. 155584-74-0
VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 37 | In Stock |
|
| 10MG | 59 | In Stock |
|
| 25MG | 112 | In Stock |
|
| 100MG | 299 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameVUF 10166
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NoteResearch use only, not for human use.
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Brief DescriptionVUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.
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DescriptionVUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAngiogenesis
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TargetEGFR
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Recptor5-HT3A| 5-HT3AB
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Research AreaInflammation/Immunology
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Indication——
Chemical Information
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CAS Number155584-74-0
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Formula Weight262.74
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Molecular FormulaC13H15ClN4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (380.60 mM)
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SMILESCN1CCN(CC1)C1=NC2=CC=CC=C2N=C1Cl
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Thompson AJ, et al. J Pharmacol Exp Ther, 2012, 341(2), 350-9.
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